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up to 1 uM
Screened for radioligand binding modulation of CNS GPCRs and toxic pharmacological off-targets at 10uM, no activity was observed.
Counter-screened against MTNR1A and was >54-fold selective for MTNR1B. Also screened against a panel of 318 GPCRs at 10uM. Secondary concentration-response assays of preliminary hits demonstrated no replicable off-target action.